Skoči na glavni sadržaj

Acta Pharmaceutica , Vol. 75 No. 2, 2025.

  • Datum izdavanja: 30.06.2025.
  • Objavljen na Hrčku: 28.06.2025.

Sadržaj

Puni tekst

Optimization of 6-(trifluoromethyl)pyrimidine derivatives as TLR8 antagonists (str. 159-183)

NIKA STRAŠEK BENEDIK, VALERIJ TALAGAYEV, TROY MATZIOL, ANA DOLŠAK, IZIDOR SOSIČ, GÜNTHER WEINDL, GERHARD WOLBER, MATEJ SOVA
Izvorni znanstveni članak


Development and evaluation of novel InhA inhibitors inspired by thiadiazole and tetrahydropyran series of inhibitors (str. 185-218)

MARTINA HRAST RAMBAHER, NINA GRADIŠEK, ROK FRLAN, IZIDOR SOSIČ, ALJOŠA BOLJE, JAKOB KLJUN, MARTIN JUHÁS, STANISLAV GOBEC, STANE PAJK
Izvorni znanstveni članak


Exploration of the chemical space of benzamide-based voltage-gated potassium channel KV1.3 inhibitors (str. 219-233)

MARZIA FOIS, ŠPELA PELCAR, JOSHUA A. NASBURG, HEIKE WULFF, LUCIJA PETERLIN MAŠIČ, TIHOMIR TOMAŠIČ
Izvorni znanstveni članak


Biochemical characteristics of the 6-nitro regioisomer of nitroxoline and its 1,2,3,4-tetrahydroquinoline analogues (str. 235-257)

ANA MITROVIĆ, DAMIJAN KNEZ, MARTINA HRAST RAMBAHER, JAKOB KLJUN, JANKO KOS, STANISLAV GOBEC, IZIDOR SOSIČ
Izvorni znanstveni članak


Impact of peroxide content in excipients and antioxidants on famotidine oxidative stability (str. 259-272)

ALEN GABRIČ, ŽIGA HODNIK, JANEZ ILAŠ, STANE PAJK
Izvorni znanstveni članak


Design, synthesis, and evaluation of a novel fluorescent probe for competitive fluorescence polarization assay to screen galectin-8 inhibitors (str. 273-282)

EDVIN PURIĆ, MARINA MARINOVIĆ, ZALA KOJEK, BARBRO KAHL-KNUTSON, HAKON LEFFLER, ULF NILSSON, MARKO ANDERLUH, JANEZ MRAVLJAK
Kratko priopćenje


α-Heteroarylthiomethyl ketones: Small molecule inhibitors of 3CLproI (str. 283-297)

DAMIJAN KNEZ, MATIC PROJ, KRIŠTOF BOZOVIČAR, STANISLAV GOBEC
Kratko priopćenje


SARS-CoV-2 structural proteins affect the expression of IL-8 and TNF-α cytokines and APOBEC genes in human lung A549 and liver Huh-7 cells (str. 299-307)

MARTINA BERGANT MARUŠIČ, MARGARIDA COSTA, ŠPELA TURK, NIKA LOVŠIN
Kratko priopćenje


Posjeta: 3.809 *